Nine of 16 stereoisomeric polyhydroxylated proline amides are potent β-N-acetylhexosaminidase inhibitors

Benjamin J. Ayers*, Andreas F.G. Glawar, R. Fernando Martínez, Nigel Ngo, Zilei Liu, George W.J. Fleet, Terry D. Butters, Robert J. Nash, Chu Yi Yu, Mark R. Wormald, Shinpei Nakagawa, Isao Adachi, Atsushi Kato, Sarah F. Jenkinson

*Corresponding author for this work

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Chemistry

Pharmacology, Toxicology and Pharmaceutical Science