@article{f7cf8e95b63e45c6a38e0cb1f72bf5ab,
title = "Synthetic Studies on a Pachastrissamine Sulfur Analogue: Synthesis of a 4-epi-Sulfur Analogue",
abstract = "A versatile synthetic procedure for a sulfur analogue of pachastrissamine (jaspine B), which involves the tandem thiolation-cyclization of a 1,4-ditosylate to construct a tetrahydrothiophene ring, was developed. Nucleophilic amino substitution of a tetrahydrothiophene-4-sulfonate with unexpected retention of the configuration afforded the sulfur analogue of 4-epi-pachastrissamine.",
keywords = "Analogue, Cyclization, Neighboring group participation, Pachastrissamine, Tetrahydrothiophene, Thiolation",
author = "Bo Liu and Kazuki Hashimoto and Hisanori Nambu and Tomoya Fujiwara and Takayuki Yakura",
note = "Publisher Copyright: {\textcopyright} 2016 The Pharmaceutical Society of Japan.",
year = "2016",
month = apr,
doi = "10.1248/cpb.c15-00996",
language = "英語",
volume = "64",
pages = "366--370",
journal = "Chemical and Pharmaceutical Bulletin",
issn = "0009-2363",
publisher = "Pharmaceutical Society of Japan",
number = "4",
}