Solution structure of epiregulin and the effect of its C-terminal domain for receptor binding affinity

Katsuharu Sato, Takashi Nakamura, Mineyuki Mizuguchi, Kazunori Miura, Masahito Tada, Tomoyasu Aizawa, Tomoharu Gomi, Kaoru Miyamoto, Keiichi Kawano*

*この論文の責任著者

研究成果: ジャーナルへの寄稿学術論文査読

17 被引用数 (Scopus)

抄録

Epiregulin (EPR), a novel member of epidermal growth factor (EGF) family, is a ligand for ErbB-1 and ErbB-4 receptors. The binding affinity of EPR for the receptors is lower than those of other EGF-family ligands. The solution structure of EPR was determined using two-dimensional nuclear magnetic resonance spectroscopy. The secondary structure in the C-terminal domain of EPR is different from other EGF-family ligands because of the lack of hydrogen bonds. The structural difference in the C-terminal domain may provide an explanation for the reduced binding affinity of EPR to the ErbB receptors.

本文言語英語
ページ(範囲)232-238
ページ数7
ジャーナルFEBS Letters
553
3
DOI
出版ステータス出版済み - 2003/10/23

ASJC Scopus 主題領域

  • 生物理学
  • 構造生物学
  • 生化学
  • 分子生物学
  • 遺伝学
  • 細胞生物学

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