A novel oxidative azidation of aromatic compounds with hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) and trimethylsilyl azide

Yasuyuki Kita; Hirofumi Tohma; Masanao Inagaki; Kenji Hatanaka; Takayuki Yakura

doi:10.1016/S0040-4039(00)92160-9

A novel oxidative azidation of aromatic compounds with hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) and trimethylsilyl azide

Yasuyuki Kita^*, Hirofumi Tohma, Masanao Inagaki, Kenji Hatanaka, Takayuki Yakura

^*Corresponding author for this work

Synthetic and Biomolecular Organic Chemistry

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Abstract

A novel and useful method for the azidation of aromatic compounds by the reaction of hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) in 1,1,1,3,3,3-hexafluoro-2-propanol followed by treatment of trimethylsilyl azide (TMSA) was developed. The possible mechanism is also discussed.

Original language	English
Pages (from-to)	4321-4324
Number of pages	4
Journal	Tetrahedron Letters
Volume	32
Issue number	34
DOIs	https://doi.org/10.1016/S0040-4039(00)92160-9
State	Published - 1991

ASJC Scopus subject areas

Biochemistry
Drug Discovery
Organic Chemistry

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title = "A novel oxidative azidation of aromatic compounds with hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) and trimethylsilyl azide",

abstract = "A novel and useful method for the azidation of aromatic compounds by the reaction of hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) in 1,1,1,3,3,3-hexafluoro-2-propanol followed by treatment of trimethylsilyl azide (TMSA) was developed. The possible mechanism is also discussed.",

author = "Yasuyuki Kita and Hirofumi Tohma and Masanao Inagaki and Kenji Hatanaka and Takayuki Yakura",

year = "1991",

doi = "10.1016/S0040-4039(00)92160-9",

language = "英語",

volume = "32",

pages = "4321--4324",

journal = "Tetrahedron Letters",

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T1 - A novel oxidative azidation of aromatic compounds with hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) and trimethylsilyl azide

AU - Kita, Yasuyuki

AU - Tohma, Hirofumi

AU - Inagaki, Masanao

AU - Hatanaka, Kenji

AU - Yakura, Takayuki

PY - 1991

Y1 - 1991

N2 - A novel and useful method for the azidation of aromatic compounds by the reaction of hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) in 1,1,1,3,3,3-hexafluoro-2-propanol followed by treatment of trimethylsilyl azide (TMSA) was developed. The possible mechanism is also discussed.

AB - A novel and useful method for the azidation of aromatic compounds by the reaction of hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) in 1,1,1,3,3,3-hexafluoro-2-propanol followed by treatment of trimethylsilyl azide (TMSA) was developed. The possible mechanism is also discussed.

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U2 - 10.1016/S0040-4039(00)92160-9

DO - 10.1016/S0040-4039(00)92160-9

M3 - 学術論文

AN - SCOPUS:0025912377

SN - 0040-4039

VL - 32

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JO - Tetrahedron Letters

JF - Tetrahedron Letters

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ER -

A novel oxidative azidation of aromatic compounds with hypervalent iodine reagent, phenyliodine(III) bis(trifluoroacetate) (PIFA) and trimethylsilyl azide

Abstract

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